284 targets, 350,097 fitting measurements and 38,916 held-out measurements. Generated from the measurement files the models were built from.
Gene symbols link to GeneCards and accessions to UniProt. The two accuracy columns are that target's own held-out accuracy, with the number of comparisons it rests on beside it. A target with few comparisons can read 0.00 or 1.00 and neither means much. Targets the model was not scored on say so.
Accuracy depends on the cutoff you are willing to act at. The figures below default to answering every comparison, which is a strength cutoff of 0.50. Raise the cutoff and accuracy rises while the number of comparisons that clear it falls, at very different rates from one target to the next.
Every column heading sorts, except endpoints. Click once for descending, again for ascending. The default is fitting measurements, largest first.
| #▾ | Gene▾ | Accession▾ | Fit measurements▾ | Fit ligands▾ | Held-out▾ | Potency accuracy▾ | Potency n▾ | Selectivity accuracy▾ | Selectivity n▾ | Endpoints |
|---|---|---|---|---|---|---|---|---|---|---|
| 1 | DRD2 | P14416 | 10,981 | 9,982 | 1,206 | 0.74 | 13,162 | 0.81 | 2,454 | Ki 8836, IC50 1100, EC50 802, Kb 152, Kd 91 |
| 2 | CNR2 | P34972 | 10,321 | 8,986 | 1,161 | 0.76 | 13,632 | 0.90 | 772 | Ki 4578, EC50 4103, IC50 1616, Kb 12, Kd 12 |
| 3 | OPRM1 | P35372 | 10,095 | 8,593 | 1,126 | 0.77 | 13,320 | 0.81 | 1,561 | Ki 5841, EC50 2405, IC50 1773, Kb 43, Kd 33 |
| 4 | CNR1 | P21554 | 9,409 | 8,284 | 1,045 | 0.79 | 12,822 | 0.90 | 785 | Ki 3703, EC50 3522, IC50 1942, Kd 168, Kb 74 |
| 5 | HCRTR2 | O43614 | 8,173 | 7,861 | 915 | 0.77 | 13,822 | 0.90 | 755 | IC50 5028, Ki 2169, EC50 800, Kd 129, Kb 47 |
| 6 | ADORA2A | P29274 | 7,979 | 7,559 | 888 | 0.76 | 9,746 | 0.83 | 1,162 | Ki 5962, IC50 1614, EC50 308, Kd 77, Kb 18 |
| 7 | OPRK1 | P41145 | 7,699 | 6,549 | 872 | 0.76 | 14,438 | 0.82 | 1,272 | Ki 4124, IC50 1849, EC50 1656, Kb 51, Kd 19 |
| 8 | HCRTR1 | O43613 | 7,307 | 6,989 | 819 | 0.79 | 10,271 | 0.89 | 757 | IC50 4800, Ki 2078, EC50 262, Kd 134, Kb 33 |
| 9 | HTR2A | P28223 | 7,215 | 6,464 | 807 | 0.73 | 14,287 | 0.79 | 2,017 | Ki 5000, IC50 1232, EC50 940, Kb 39, Kd 4 |
| 10 | OPRD1 | P41143 | 6,982 | 5,819 | 767 | 0.78 | 13,565 | 0.88 | 1,167 | Ki 4148, EC50 1439, IC50 1316, Kd 41, Kb 38 |
| 11 | DRD3 | P35462 | 6,642 | 6,074 | 755 | 0.75 | 7,795 | 0.78 | 1,896 | Ki 5700, EC50 493, IC50 396, Kb 30, Kd 23 |
| 12 | HTR1A | P08908 | 6,488 | 5,868 | 715 | 0.73 | 10,716 | 0.76 | 1,670 | Ki 4894, EC50 836, IC50 650, Kd 60, Kb 48 |
| 13 | ADORA1 | P30542 | 6,082 | 5,699 | 681 | 0.73 | 8,500 | 0.83 | 1,052 | Ki 4733, IC50 757, EC50 434, Kd 150, Kb 8 |
| 14 | ADORA3 | P0DMS8 | 5,971 | 5,480 | 670 | 0.76 | 8,378 | 0.82 | 1,069 | Ki 4714, IC50 907, EC50 250, Kd 68, Kb 32 |
| 15 | PTGDR2 | Q9Y5Y4 | 5,951 | 5,629 | 652 | 0.73 | 9,504 | 0.95 | 65 | IC50 3661, Ki 1725, EC50 554, Kb 6, Kd 5 |
| 16 | HTR6 | P50406 | 5,133 | 4,343 | 567 | 0.76 | 9,395 | 0.74 | 1,001 | Ki 3769, IC50 887, Kb 272, EC50 135, Kd 70 |
| 17 | HRH3 | Q9Y5N1 | 5,053 | 4,300 | 547 | 0.74 | 8,036 | 0.84 | 279 | Ki 3664, IC50 727, EC50 339, Kd 251, Kb 72 |
| 18 | HTR2C | P28335 | 4,788 | 4,276 | 538 | 0.72 | 13,774 | 0.80 | 1,522 | Ki 2712, EC50 1061, IC50 1005, Kb 8, Kd 2 |
| 19 | ADORA2B | P29275 | 4,745 | 4,532 | 519 | 0.80 | 9,518 | 0.91 | 719 | Ki 2536, IC50 1744, EC50 385, Kb 43, Kd 37 |
| 20 | LPAR1 | Q92633 | 4,522 | 4,396 | 507 | 0.71 | 5,546 | 0.83 | 36 | IC50 3903, EC50 449, Ki 125, Kb 39, Kd 6 |
| 21 | MC4R | P32245 | 4,371 | 3,393 | 474 | 0.79 | 14,362 | 0.80 | 446 | Ki 1852, EC50 1454, IC50 1025, Kd 27, Kb 13 |
| 22 | CRHR1 | P34998 | 4,065 | 3,826 | 452 | 0.78 | 5,053 | 0.82 | 11 | IC50 2487, Ki 1465, EC50 93, Kd 20 |
| 23 | S1PR1 | P21453 | 3,912 | 3,556 | 441 | 0.77 | 9,356 | 0.94 | 384 | EC50 2502, IC50 1271, Ki 129, Kd 9, Kb 1 |
| 24 | MCHR1 | Q99705 | 3,910 | 3,667 | 438 | 0.73 | 9,805 | 0.82 | 57 | IC50 2306, Ki 1483, EC50 61, Kb 57, Kd 3 |
| 25 | GRM5 | P41594 | 3,628 | 3,186 | 410 | 0.75 | 10,951 | 0.84 | 88 | IC50 1894, EC50 1198, Ki 525, Kb 9, Kd 2 |
| 26 | DRD4 | P21917 | 3,496 | 3,059 | 385 | 0.72 | 6,486 | 0.80 | 1,080 | Ki 2758, IC50 369, EC50 354, Kd 12, Kb 3 |
| 27 | CHRM1 | P11229 | 3,464 | 3,249 | 392 | 0.74 | 13,884 | 0.75 | 903 | Ki 1501, EC50 886, IC50 860, Kb 148, Kd 69 |
| 28 | APLNR | P35414 | 3,358 | 3,196 | 371 | 0.73 | 5,253 | 0.66 | 44 | EC50 2984, Ki 240, IC50 133, Kd 1 |
| 29 | HTR7 | P34969 | 3,345 | 3,165 | 367 | 0.73 | 6,294 | 0.76 | 1,025 | Ki 2631, IC50 416, EC50 231, Kb 58, Kd 9 |
| 30 | GLP1R | P43220 | 3,099 | 2,924 | 345 | 0.81 | 4,917 | 0.78 | 76 | EC50 2813, IC50 231, Ki 45, Kd 10 |
| 31 | OPRL1 | P41146 | 3,084 | 2,684 | 342 | 0.76 | 7,832 | 0.90 | 370 | Ki 2003, IC50 647, EC50 372, Kb 51, Kd 11 |
| 32 | CHRM3 | P20309 | 3,083 | 2,897 | 348 | 0.82 | 9,197 | 0.76 | 859 | Ki 1887, IC50 942, EC50 167, Kd 87 |
| 33 | HRH4 | Q9H3N8 | 3,062 | 2,697 | 331 | 0.75 | 5,427 | 0.85 | 215 | Ki 1673, EC50 1014, IC50 188, Kd 131, Kb 56 |
| 34 | MRGPRX2 | Q96LB1 | 2,811 | 2,785 | 313 | 0.83 | 2,727 | 1.00 | 4 | IC50 2496, EC50 289, Kd 26 |
| 35 | CHRM2 | P08172 | 2,787 | 2,532 | 317 | 0.80 | 8,180 | 0.78 | 853 | Ki 1598, IC50 601, EC50 272, Kb 178, Kd 138 |
| 36 | HRH1 | P35367 | 2,784 | 2,615 | 313 | 0.77 | 5,676 | 0.76 | 769 | Ki 1506, EC50 664, IC50 391, Kd 164, Kb 59 |
| 37 | ADRB2 | P07550 | 2,728 | 2,358 | 300 | 0.81 | 10,065 | 0.77 | 476 | EC50 1217, IC50 675, Ki 665, Kd 169, Kb 2 |
| 38 | TACR1 | P25103 | 2,616 | 2,495 | 293 | 0.80 | 9,339 | 0.78 | 162 | IC50 1643, Ki 860, Kd 96, EC50 15, Kb 2 |
| 39 | HTR2B | P41595 | 2,565 | 2,169 | 288 | 0.74 | 7,208 | 0.74 | 1,146 | Ki 1669, EC50 526, IC50 345, Kb 24, Kd 1 |
| 40 | FFAR1 | O14842 | 2,550 | 2,399 | 284 | 0.72 | 4,832 | 0.94 | 32 | EC50 2320, Ki 126, IC50 94, Kd 10 |
| 41 | S1PR3 | Q99500 | 2,450 | 2,411 | 272 | 0.83 | 5,946 | 0.94 | 359 | EC50 1617, IC50 820, Kd 8, Ki 5 |
| 42 | GHSR | Q92847 | 2,346 | 1,925 | 261 | 0.72 | 10,462 | 0.86 | 7 | IC50 879, EC50 792, Ki 603, Kb 69, Kd 3 |
| 43 | CHRM4 | P08173 | 2,302 | 2,159 | 259 | 0.77 | 7,945 | 0.78 | 691 | Ki 1312, EC50 656, IC50 300, Kb 27, Kd 7 |
| 44 | CCR5 | P51681 | 2,261 | 2,230 | 257 | 0.77 | 5,073 | 0.73 | 56 | IC50 2050, Ki 142, EC50 55, Kd 14 |
| 45 | FPR2 | P25090 | 2,154 | 2,097 | 237 | 0.78 | 6,969 | 0.86 | 86 | EC50 1326, IC50 462, Kd 339, Ki 27 |
| 46 | GRM2 | Q14416 | 2,122 | 1,895 | 228 | 0.76 | 9,884 | 0.69 | 72 | EC50 939, IC50 921, Ki 205, Kd 44, Kb 13 |
| 47 | CCR2 | P41597 | 2,070 | 1,985 | 227 | 0.73 | 5,135 | 0.95 | 21 | IC50 1754, Ki 290, Kd 17, EC50 9 |
| 48 | ADRA1A | P35348 | 2,044 | 1,931 | 224 | 0.80 | 5,757 | 0.83 | 774 | Ki 1414, IC50 309, EC50 290, Kd 18, Kb 13 |
| 49 | CHRM5 | P08912 | 2,023 | 1,935 | 225 | 0.75 | 8,314 | 0.75 | 621 | IC50 911, Ki 896, EC50 213, Kd 3 |
| 50 | AVPR1A | P37288 | 1,978 | 1,691 | 220 | 0.78 | 7,201 | 0.83 | 224 | Ki 1049, IC50 690, EC50 214, Kb 17, Kd 8 |
| 51 | DRD1 | P21728 | 1,947 | 1,750 | 214 | 0.76 | 5,346 | 0.75 | 782 | Ki 1423, EC50 265, IC50 218, Kd 30, Kb 11 |
| 52 | ADRB1 | P08588 | 1,849 | 1,709 | 204 | 0.78 | 6,250 | 0.81 | 527 | EC50 760, IC50 588, Ki 403, Kd 97, Kb 1 |
| 53 | GPR17 | Q13304 | 1,826 | 1,813 | 207 | 0.79 | 3,093 | 0.69 | 16 | IC50 1532, Kb 212, EC50 67, Ki 14, Kd 1 |
| 54 | GPR119 | Q8TDV5 | 1,737 | 1,678 | 190 | 0.74 | 4,661 | 0.50 | 24 | EC50 1656, Ki 47, IC50 34 |
| 55 | CXCR3 | P49682 | 1,709 | 1,679 | 189 | 0.76 | 5,246 | 0.47 | 19 | IC50 1405, Ki 266, EC50 34, Kd 4 |
| 56 | CCKBR | P32239 | 1,696 | 1,553 | 179 | 0.82 | 6,262 | 0.85 | 47 | IC50 1131, Ki 452, EC50 106, Kd 7 |
| 57 | ADRA1B | P35368 | 1,688 | 1,616 | 184 | 0.76 | 4,812 | 0.78 | 613 | Ki 1310, EC50 213, IC50 150, Kd 10, Kb 5 |
| 58 | GRM4 | Q14833 | 1,655 | 1,600 | 190 | 0.77 | 4,972 | 0.78 | 79 | EC50 1487, IC50 85, Ki 70, Kb 13 |
| 59 | ADRB3 | P13945 | 1,653 | 1,539 | 188 | 0.74 | 5,631 | 0.79 | 392 | EC50 1174, Ki 340, IC50 82, Kd 57 |
| 60 | P2RY1 | P47900 | 1,617 | 1,142 | 181 | 0.70 | 4,360 | 0.71 | 14 | Ki 961, IC50 587, EC50 62, Kd 6, Kb 1 |
| 61 | GNRHR | P30968 | 1,614 | 1,515 | 179 | 0.78 | 7,002 | 1.00 | 2 | IC50 912, Ki 664, Kd 35, EC50 2, Kb 1 |
| 62 | EDNRA | P25101 | 1,585 | 1,516 | 173 | 0.80 | 5,079 | 0.70 | 178 | IC50 1278, Ki 227, Kb 65, EC50 11, Kd 4 |
| 63 | SSTR4 | P31391 | 1,584 | 1,336 | 180 | 0.76 | 5,308 | 0.82 | 253 | EC50 604, IC50 532, Ki 418, Kd 30 |
| 64 | HTR1D | P28221 | 1,569 | 1,383 | 171 | 0.80 | 5,674 | 0.77 | 597 | Ki 1081, IC50 310, EC50 166, Kb 9, Kd 3 |
| 65 | ADRA1D | P25100 | 1,567 | 1,433 | 170 | 0.75 | 4,888 | 0.80 | 605 | Ki 1139, IC50 219, EC50 204, Kb 5 |
| 66 | MC1R | Q01726 | 1,549 | 1,095 | 166 | 0.81 | 4,922 | 0.83 | 249 | EC50 737, Ki 482, IC50 326, Kd 4 |
| 67 | MC5R | P33032 | 1,516 | 1,269 | 167 | 0.83 | 2,706 | 0.76 | 257 | IC50 771, Ki 421, EC50 320, Kd 4 |
| 68 | PTGER4 | P35408 | 1,498 | 1,265 | 166 | 0.79 | 4,643 | 0.93 | 187 | IC50 661, Ki 534, EC50 252, Kb 44, Kd 7 |
| 69 | MC3R | P41968 | 1,497 | 1,075 | 160 | 0.81 | 4,176 | 0.83 | 355 | Ki 607, EC50 502, IC50 368, Kd 20 |
| 70 | GCGR | P47871 | 1,476 | 1,420 | 166 | 0.80 | 4,725 | 0.88 | 48 | IC50 782, EC50 372, Ki 273, Kb 49 |
| 71 | SSTR2 | P30874 | 1,461 | 1,427 | 163 | 0.85 | 3,133 | 0.82 | 240 | Ki 526, IC50 457, EC50 443, Kd 35 |
| 72 | AGTR1 | P30556 | 1,458 | 1,407 | 164 | 0.86 | 4,984 | 0.67 | 121 | IC50 1062, Ki 200, EC50 164, Kd 24, Kb 8 |
| 73 | ADRA2A | P08913 | 1,442 | 1,178 | 162 | 0.78 | 5,387 | 0.74 | 811 | Ki 910, IC50 273, EC50 186, Kb 67, Kd 6 |
| 74 | ACKR3 | P25106 | 1,433 | 1,417 | 162 | 0.75 | 5,068 | 1.00 | 12 | IC50 722, EC50 625, Ki 83, Kd 3 |
| 75 | HTR1B | P28222 | 1,417 | 1,319 | 156 | 0.80 | 5,174 | 0.79 | 551 | Ki 1013, IC50 280, EC50 111, Kd 7, Kb 6 |
| 76 | FFAR4 | Q5NUL3 | 1,412 | 1,410 | 157 | 0.78 | 4,165 | 0.88 | 43 | EC50 1400, IC50 12 |
| 77 | TACR3 | P29371 | 1,403 | 1,159 | 156 | 0.79 | 4,502 | 0.78 | 98 | Ki 806, IC50 463, EC50 114, Kb 10, Kd 10 |
| 78 | P2RY12 | Q9H244 | 1,383 | 1,208 | 159 | 0.77 | 4,977 | 0.80 | 5 | IC50 701, Ki 607, EC50 68, Kb 4, Kd 3 |
| 79 | CXCR2 | P25025 | 1,329 | 1,291 | 154 | 0.77 | 4,478 | 0.84 | 91 | IC50 1094, Ki 215, Kd 18, EC50 2 |
| 80 | CXCR4 | P61073 | 1,319 | 1,200 | 149 | 0.71 | 4,793 | 0.85 | 27 | IC50 1094, EC50 204, Ki 13, Kb 4, Kd 4 |
| 81 | NPY5R | Q15761 | 1,313 | 1,246 | 143 | 0.75 | 4,650 | 0.93 | 55 | IC50 714, Ki 563, EC50 32, Kb 4 |
| 82 | NPY1R | P25929 | 1,303 | 1,178 | 141 | 0.81 | 3,377 | 0.70 | 124 | Ki 602, IC50 481, EC50 142, Kb 58, Kd 20 |
| 83 | MTNR1A | P48039 | 1,288 | 1,097 | 145 | 0.79 | 4,728 | 0.74 | 157 | Ki 891, IC50 204, EC50 168, Kb 23, Kd 2 |
| 84 | OXTR | P30559 | 1,242 | 1,124 | 132 | 0.80 | 3,208 | 0.87 | 138 | Ki 635, EC50 360, IC50 214, Kd 33 |
| 85 | CRHR2 | Q13324 | 1,233 | 1,228 | 137 | 1.00 | 280 | 0.88 | 8 | IC50 1219, Ki 9, EC50 5 |
| 86 | TBXA2R | P21731 | 1,219 | 1,178 | 138 | 0.83 | 2,989 | 0.88 | 96 | IC50 560, Ki 412, Kd 204, EC50 41, Kb 2 |
| 87 | F2RL3 | Q96RI0 | 1,218 | 1,132 | 133 | 0.79 | 4,492 | 1.00 | 7 | IC50 793, EC50 422, Kd 3 |
| 88 | GPBAR1 | Q8TDU6 | 1,198 | 1,194 | 133 | 0.72 | 4,833 | 0.00 | 1 | EC50 1166, IC50 32 |
| 89 | EDNRB | P24530 | 1,169 | 1,140 | 127 | 0.82 | 4,832 | 0.86 | 118 | IC50 981, Ki 177, Kd 5, Kb 4, EC50 2 |
| 90 | CALCRL | Q16602 | 1,152 | 820 | 133 | 0.85 | 4,158 | not scored | Ki 580, IC50 547, EC50 12, Kd 7, Kb 6 | |
| 91 | MTNR1B | P49286 | 1,145 | 960 | 137 | 0.77 | 4,620 | 0.84 | 121 | Ki 858, EC50 165, IC50 86, Kb 33, Kd 3 |
| 92 | SSTR3 | P32745 | 1,138 | 978 | 128 | 0.84 | 2,310 | 0.80 | 228 | IC50 531, Ki 361, EC50 176, Kd 70 |
| 93 | GRM1 | Q13255 | 1,138 | 1,040 | 129 | 0.84 | 3,804 | 0.82 | 102 | IC50 781, EC50 255, Ki 88, Kb 14 |
| 94 | SSTR5 | P35346 | 1,129 | 1,086 | 126 | 0.85 | 3,310 | 0.85 | 239 | IC50 668, Ki 360, EC50 68, Kd 33 |
| 95 | C5AR1 | P21730 | 1,125 | 1,102 | 129 | 0.82 | 4,491 | 0.60 | 5 | IC50 1022, EC50 49, Ki 41, Kb 10, Kd 3 |
| 96 | PTGER3 | P43115 | 1,118 | 967 | 119 | 0.83 | 2,501 | 0.87 | 121 | IC50 501, Ki 485, EC50 121, Kb 11 |
| 97 | TAAR1 | Q96RJ0 | 1,113 | 699 | 127 | 0.62 | 3,845 | 1.00 | 1 | EC50 659, IC50 408, Ki 46 |
| 98 | AVPR2 | P30518 | 1,107 | 1,038 | 123 | 0.82 | 2,534 | 0.84 | 167 | Ki 470, IC50 367, EC50 261, Kd 9 |
| 99 | TACR2 | P21452 | 1,105 | 1,043 | 124 | 0.87 | 3,937 | 0.65 | 267 | Ki 805, IC50 285, Kd 9, EC50 5, Kb 1 |
| 100 | NPY2R | P49146 | 1,098 | 979 | 121 | 0.90 | 2,520 | 0.71 | 111 | IC50 532, Ki 279, EC50 271, Kd 15, Kb 1 |
| 101 | PTGER2 | P43116 | 1,081 | 968 | 117 | 0.81 | 1,682 | 0.90 | 157 | Ki 380, EC50 323, IC50 196, Kb 175, Kd 7 |
| 102 | CCR3 | P51677 | 1,069 | 1,059 | 118 | 0.82 | 3,936 | 0.91 | 22 | IC50 686, Ki 373, EC50 5, Kb 3, Kd 2 |
| 103 | ADRA2C | P18825 | 1,064 | 821 | 121 | 0.71 | 3,349 | 0.73 | 727 | Ki 705, EC50 148, IC50 140, Kb 70, Kd 1 |
| 104 | PTGER1 | P34995 | 1,044 | 923 | 121 | 0.79 | 2,993 | 0.85 | 101 | IC50 607, Ki 371, EC50 42, Kd 14, Kb 10 |
| 105 | BDKRB1 | P46663 | 1,041 | 805 | 114 | 0.74 | 3,073 | 0.78 | 9 | Ki 637, IC50 398, Kd 2, Kb 2, EC50 2 |
| 106 | GPR6 | P46095 | 1,040 | 1,035 | 117 | 0.81 | 3,545 | 1.00 | 10 | IC50 675, EC50 360, Ki 4, Kd 1 |
| 107 | FPR1 | P21462 | 1,006 | 975 | 110 | 0.71 | 1,944 | 0.84 | 63 | EC50 503, Ki 255, IC50 206, Kd 42 |
| 108 | F2R | P25116 | 962 | 910 | 110 | 0.82 | 3,776 | 1.00 | 6 | IC50 780, EC50 95, Ki 73, Kd 14 |
| 109 | HTR4 | Q13639 | 947 | 758 | 100 | 0.78 | 2,201 | 0.86 | 101 | Ki 459, EC50 386, IC50 87, Kb 12, Kd 3 |
| 110 | GPR55 | Q9Y2T6 | 938 | 879 | 108 | 0.79 | 2,567 | 0.76 | 72 | IC50 557, EC50 374, Kb 4, Kd 3 |
| 111 | GPR84 | Q9NQS5 | 907 | 843 | 102 | 0.79 | 2,339 | not scored | IC50 564, EC50 267, Ki 70, Kd 4, Kb 2 | |
| 112 | HRH2 | P25021 | 905 | 744 | 99 | 0.82 | 1,551 | 0.74 | 449 | Ki 574, EC50 136, IC50 118, Kd 60, Kb 17 |
| 113 | S1PR2 | O95136 | 904 | 888 | 102 | 0.90 | 1,477 | 0.88 | 142 | IC50 611, EC50 226, Kd 66, Ki 1 |
| 114 | CCR4 | P51679 | 891 | 821 | 96 | 0.83 | 2,479 | 0.75 | 12 | IC50 751, Ki 90, Kd 41, EC50 9 |
| 115 | CCR1 | P32246 | 889 | 842 | 96 | 0.78 | 3,094 | 0.80 | 55 | IC50 722, Ki 148, EC50 18, Kd 1 |
| 116 | ADRA2B | P18089 | 884 | 688 | 101 | 0.68 | 2,217 | 0.71 | 673 | Ki 603, IC50 160, EC50 84, Kb 36, Kd 1 |
| 117 | GPR35 | Q9HC97 | 882 | 570 | 99 | 0.85 | 1,621 | 0.83 | 66 | EC50 422, IC50 400, Ki 56, Kd 4 |
| 118 | PTGDR | Q13258 | 881 | 796 | 91 | 0.88 | 1,245 | 0.92 | 128 | IC50 440, Ki 325, Kb 58, EC50 57, Kd 1 |
| 119 | CCR6 | P51684 | 863 | 859 | 98 | 0.88 | 4,018 | 0.76 | 21 | IC50 858, Ki 4, EC50 1 |
| 120 | HCAR2 | Q8TDS4 | 855 | 663 | 98 | 0.82 | 2,462 | 0.83 | 12 | EC50 562, IC50 261, Ki 32 |
| 121 | AVPR1B | P47901 | 815 | 805 | 92 | 0.86 | 1,461 | 0.95 | 116 | IC50 395, Ki 223, EC50 192, Kd 5 |
| 122 | SSTR1 | P30872 | 807 | 797 | 90 | 0.86 | 1,325 | 0.88 | 232 | IC50 504, Ki 238, Kd 50, EC50 15 |
| 123 | NTSR1 | P30989 | 791 | 699 | 80 | 0.76 | 1,281 | 0.66 | 59 | EC50 511, Ki 152, IC50 115, Kd 13 |
| 124 | FFAR2 | O15552 | 790 | 768 | 87 | 0.74 | 1,657 | 1.00 | 4 | EC50 588, IC50 178, Ki 24 |
| 125 | S1PR4 | O95977 | 789 | 778 | 88 | 0.81 | 1,661 | 0.87 | 161 | IC50 439, EC50 339, Kd 8, Ki 2, Kb 1 |
| 126 | SMO | Q99835 | 775 | 752 | 88 | 0.79 | 3,129 | not scored | IC50 729, EC50 21, Ki 20, Kd 5 | |
| 127 | AGTR2 | P50052 | 761 | 752 | 85 | 0.80 | 2,216 | 0.98 | 41 | IC50 544, Ki 217 |
| 128 | HTR5A | P47898 | 741 | 707 | 81 | 0.84 | 1,341 | 0.78 | 403 | Ki 451, EC50 242, IC50 46, Kd 2 |
| 129 | UTS2R | Q9UKP6 | 694 | 618 | 74 | 0.80 | 826 | not scored | Ki 292, EC50 218, IC50 179, Kd 5 | |
| 130 | CCKAR | P32238 | 686 | 470 | 69 | 0.87 | 724 | 0.79 | 80 | IC50 318, EC50 191, Ki 176, Kd 1 |
| 131 | PTGIR | P43119 | 628 | 583 | 70 | 0.79 | 507 | 0.87 | 70 | Ki 256, IC50 166, EC50 162, Kb 44 |
| 132 | PTAFR | P25105 | 625 | 616 | 68 | 0.80 | 2,018 | 1.00 | 1 | IC50 602, Ki 22, Kd 1 |
| 133 | BDKRB2 | P30411 | 625 | 537 | 69 | 0.84 | 858 | 0.73 | 45 | Ki 303, IC50 225, Kd 95, EC50 2 |
| 134 | S1PR5 | Q9H228 | 619 | 605 | 68 | 0.78 | 1,129 | 0.82 | 151 | EC50 354, IC50 252, Kd 8, Ki 5 |
| 135 | DRD5 | P21918 | 594 | 581 | 66 | 0.81 | 1,452 | 0.80 | 379 | Ki 533, EC50 40, IC50 18, Kd 3 |
| 136 | CX3CR1 | P49238 | 594 | 589 | 65 | 0.80 | 1,152 | 0.74 | 38 | IC50 469, EC50 70, Ki 55 |
| 137 | CASR | P41180 | 592 | 591 | 66 | 0.80 | 1,067 | 1.00 | 1 | IC50 360, EC50 232 |
| 138 | PTGFR | P43088 | 567 | 555 | 63 | 0.83 | 1,129 | 0.91 | 58 | IC50 418, Ki 86, EC50 61, Kb 2 |
| 139 | MLNR | O43193 | 548 | 484 | 64 | 0.70 | 608 | 1.00 | 3 | EC50 290, Ki 160, IC50 98 |
| 140 | LTB4R | Q15722 | 530 | 491 | 59 | 0.77 | 542 | not scored | IC50 249, EC50 152, Ki 123, Kb 5, Kd 1 | |
| 141 | BRS3 | P32247 | 527 | 363 | 53 | 0.79 | 704 | 0.71 | 7 | EC50 328, IC50 178, Ki 21 |
| 142 | NPBWR1 | P48145 | 506 | 499 | 56 | 0.83 | 1,275 | 0.67 | 24 | IC50 460, EC50 46 |
| 143 | CALCR | P30988 | 480 | 355 | 48 | 0.86 | 703 | not scored | EC50 342, IC50 125, Ki 13 | |
| 144 | GPR183 | P32249 | 464 | 463 | 52 | 0.82 | 1,089 | 0.63 | 30 | IC50 455, EC50 8, Kd 1 |
| 145 | FPR3 | P25089 | 456 | 456 | 51 | 0.87 | 1,017 | 0.80 | 66 | EC50 419, IC50 37 |
| 146 | GPR88 | Q9GZN0 | 449 | 444 | 49 | 0.80 | 1,162 | not scored | EC50 443, Ki 5, Kd 1 | |
| 147 | P2RY2 | P41231 | 442 | 434 | 50 | 0.76 | 424 | 0.73 | 40 | EC50 248, IC50 132, Kd 40, Ki 22 |
| 148 | NPY4R | P50391 | 431 | 275 | 52 | 0.84 | 425 | 0.91 | 55 | Ki 215, EC50 135, IC50 44, Kb 32, Kd 5 |
| 149 | GPR139 | Q6DWJ6 | 420 | 336 | 44 | 0.79 | 592 | not scored | EC50 334, Ki 86 | |
| 150 | CMKLR1 | Q99788 | 415 | 385 | 46 | 0.91 | 257 | 1.00 | 3 | IC50 332, EC50 82, Ki 1 |
| 151 | GIPR | P48546 | 406 | 405 | 45 | 0.84 | 237 | 0.87 | 30 | EC50 263, IC50 140, Ki 3 |
| 152 | P2RY14 | Q15391 | 404 | 377 | 46 | 0.78 | 488 | 0.88 | 17 | IC50 321, EC50 47, Ki 31, Kd 4, Kb 1 |
| 153 | CXCR1 | P25024 | 386 | 377 | 42 | 0.83 | 359 | 1.00 | 37 | IC50 290, Ki 91, Kd 4, EC50 1 |
| 154 | P2RY6 | Q15077 | 375 | 373 | 42 | 0.74 | 424 | 0.64 | 33 | EC50 252, IC50 115, Ki 6, Kd 2 |
| 155 | LPAR2 | Q9HBW0 | 367 | 362 | 41 | 0.87 | 372 | 0.84 | 32 | IC50 299, EC50 61, Ki 7 |
| 156 | CCR9 | P51686 | 359 | 357 | 40 | 0.89 | 159 | not scored | IC50 237, Ki 121, EC50 1 | |
| 157 | KISS1R | Q969F8 | 357 | 284 | 44 | 0.82 | 362 | 1.00 | 4 | EC50 186, IC50 94, Ki 77 |
| 158 | GPR52 | Q9Y2T5 | 332 | 332 | 37 | 0.86 | 486 | not scored | EC50 308, IC50 24 | |
| 159 | GRM3 | Q14832 | 329 | 242 | 39 | 0.79 | 223 | 0.71 | 58 | IC50 144, EC50 109, Ki 76 |
| 160 | PRLHR | P49683 | 314 | 231 | 35 | 0.80 | 204 | not scored | Ki 144, IC50 86, EC50 84 | |
| 161 | HTR1E | P28566 | 309 | 287 | 35 | 0.86 | 176 | 0.84 | 282 | Ki 237, IC50 40, EC50 32 |
| 162 | GRM7 | Q14831 | 302 | 288 | 33 | 0.79 | 123 | 0.97 | 35 | IC50 163, EC50 122, Ki 17 |
| 163 | PTH1R | Q03431 | 298 | 282 | 32 | 0.88 | 199 | not scored | EC50 213, IC50 55, Ki 24, Kd 6 | |
| 164 | TAS2R8 | Q9NYW2 | 290 | 290 | 32 | 0.82 | 491 | not scored | IC50 289, EC50 1 | |
| 165 | PROKR1 | Q8TCW9 | 282 | 282 | 31 | 0.69 | 463 | not scored | IC50 279, Ki 3 | |
| 166 | CXCR6 | O00574 | 280 | 278 | 31 | 0.94 | 212 | not scored | IC50 278, EC50 1, Kd 1 | |
| 167 | MRGPRX4 | Q96LA9 | 278 | 278 | 31 | 0.79 | 248 | not scored | IC50 278 | |
| 168 | LPAR3 | Q9UBY5 | 271 | 232 | 28 | 0.81 | 140 | 0.75 | 20 | IC50 147, EC50 65, Ki 59 |
| 169 | C3AR1 | Q16581 | 261 | 207 | 29 | 0.63 | 205 | 0.75 | 4 | IC50 162, EC50 98, Kd 1 |
| 170 | CYSLTR1 | Q9Y271 | 250 | 241 | 30 | 0.84 | 278 | 0.42 | 38 | IC50 217, Ki 12, EC50 12, Kd 9 |
| 171 | CCR8 | P51685 | 246 | 236 | 27 | 0.76 | 172 | 0.25 | 4 | IC50 162, Ki 68, EC50 16 |
| 172 | GRPR | P30550 | 240 | 232 | 26 | 0.83 | 248 | 0.71 | 7 | IC50 184, Ki 47, EC50 8, Kb 1 |
| 173 | GALR3 | O60755 | 239 | 239 | 26 | 0.64 | 220 | not scored | IC50 211, Ki 24, Kd 4 | |
| 174 | GPR18 | Q14330 | 238 | 190 | 29 | 0.90 | 134 | 0.89 | 18 | IC50 128, EC50 108, Kd 1, Kb 1 |
| 175 | P2RY4 | P51582 | 229 | 228 | 25 | 0.83 | 139 | 0.74 | 31 | EC50 148, IC50 80, Kb 1 |
| 176 | RXFP1 | Q9HBX9 | 229 | 226 | 25 | 0.82 | 297 | 1.00 | 2 | EC50 218, IC50 6, Ki 5 |
| 177 | F2RL1 | P55085 | 218 | 216 | 25 | 0.60 | 124 | 1.00 | 1 | EC50 113, IC50 103, Ki 2 |
| 178 | NPFFR2 | Q9Y5X5 | 201 | 175 | 20 | 0.82 | 126 | 0.84 | 32 | Ki 120, EC50 66, IC50 8, Kd 7 |
| 179 | GPR142 | Q7Z601 | 199 | 199 | 22 | 0.77 | 149 | not scored | EC50 156, IC50 43 | |
| 180 | HTR1F | P30939 | 198 | 172 | 19 | 0.62 | 58 | 0.76 | 109 | Ki 125, EC50 59, IC50 14 |
| 181 | GRM8 | O00222 | 196 | 186 | 23 | 0.73 | 91 | 0.87 | 53 | EC50 134, IC50 42, Ki 19, Kd 1 |
| 182 | NTSR2 | O95665 | 194 | 184 | 20 | 0.64 | 72 | 0.88 | 16 | Ki 116, EC50 49, IC50 26, Kd 3 |
| 183 | GPR3 | P46089 | 187 | 184 | 20 | 0.79 | 78 | 1.00 | 10 | IC50 142, EC50 43, Kd 1, Ki 1 |
| 184 | NPFFR1 | Q9GZQ6 | 184 | 160 | 21 | 0.74 | 108 | 0.88 | 25 | Ki 116, EC50 50, Kd 9, IC50 8, Kb 1 |
| 185 | HCAR1 | Q9BXC0 | 180 | 180 | 20 | 0.77 | 111 | 1.00 | 2 | EC50 180 |
| 186 | NMBR | P28336 | 174 | 167 | 19 | 0.81 | 59 | 0.67 | 6 | Ki 100, IC50 64, EC50 8, Kb 2 |
| 187 | NMUR2 | Q9GZQ4 | 163 | 119 | 17 | 0.79 | 72 | 0.69 | 13 | EC50 113, IC50 43, Ki 3, Kd 2, Kb 2 |
| 188 | ADCYAP1R1 | P41586 | 162 | 95 | 18 | 0.83 | 60 | 0.00 | 2 | IC50 79, EC50 65, Ki 15, Kd 3 |
| 189 | QRFPR | Q96P65 | 161 | 128 | 16 | 0.86 | 49 | 1.00 | 2 | EC50 85, IC50 71, Ki 5 |
| 190 | GRM6 | O15303 | 157 | 148 | 18 | 0.76 | 71 | 0.86 | 42 | EC50 98, IC50 36, Ki 23 |
| 191 | LPAR5 | Q9H1C0 | 157 | 156 | 17 | 0.85 | 130 | 0.73 | 11 | IC50 142, EC50 14, Ki 1 |
| 192 | MRGPRX1 | Q96LB2 | 144 | 144 | 16 | 0.81 | 63 | 1.00 | 2 | EC50 117, IC50 27 |
| 193 | MCHR2 | Q969V1 | 142 | 141 | 16 | 0.85 | 34 | 0.89 | 9 | Ki 86, IC50 56 |
| 194 | RXFP3 | Q9NSD7 | 142 | 118 | 16 | 0.86 | 36 | 0.67 | 6 | EC50 66, IC50 41, Ki 35 |
| 195 | CCRL2 | O00421 | 140 | 140 | 16 | 0.76 | 119 | 1.00 | 1 | IC50 140 |
| 196 | TAS2R14 | Q9NYV8 | 139 | 138 | 15 | 0.77 | 69 | not scored | IC50 105, EC50 34 | |
| 197 | GPR34 | Q9UPC5 | 133 | 133 | 15 | 1.00 | 13 | 1.00 | 3 | IC50 93, EC50 40 |
| 198 | NMUR1 | Q9HB89 | 131 | 90 | 14 | 0.81 | 42 | 0.69 | 13 | EC50 81, IC50 43, Ki 3, Kd 2, Kb 2 |
| 199 | GALR2 | O43603 | 128 | 125 | 14 | 0.58 | 43 | 0.64 | 44 | IC50 78, Ki 32, EC50 11, Kd 7 |
| 200 | HCAR3 | P49019 | 114 | 113 | 13 | 0.85 | 75 | 0.75 | 8 | EC50 110, IC50 4 |
| 201 | FSHR | P23945 | 111 | 111 | 12 | 0.69 | 32 | 1.00 | 3 | EC50 56, IC50 55 |
| 202 | GPER1 | Q99527 | 109 | 105 | 13 | 0.29 | 28 | 0.00 | 1 | IC50 100, EC50 5, Ki 3, Kd 1 |
| 203 | GLP2R | O95838 | 108 | 108 | 12 | 0.80 | 55 | 0.92 | 12 | EC50 100, IC50 8 |
| 204 | LTB4R2 | Q9NPC1 | 108 | 99 | 11 | 0.84 | 45 | not scored | EC50 67, IC50 37, Kd 3, Ki 1 | |
| 205 | CYSLTR2 | Q9NS75 | 108 | 105 | 12 | 0.88 | 52 | 0.83 | 24 | IC50 97, EC50 10, Ki 1 |
| 206 | GPR65 | Q8IYL9 | 106 | 106 | 12 | 0.89 | 45 | 0.74 | 23 | IC50 103, EC50 3 |
| 207 | SUCNR1 | Q9BXA5 | 101 | 91 | 11 | 0.71 | 24 | 1.00 | 1 | IC50 70, EC50 19, Ki 9, Kd 3 |
| 208 | GALR1 | P47211 | 99 | 95 | 11 | 0.72 | 25 | 0.75 | 8 | IC50 58, Ki 34, Kd 7 |
| 209 | GPR174 | Q9BXC1 | 93 | 88 | 11 | 0.69 | 32 | 0.80 | 5 | EC50 88, IC50 5 |
| 210 | CXCR5 | P32302 | 89 | 88 | 10 | 0.78 | 45 | 0.38 | 8 | IC50 87, EC50 2 |
| 211 | FFAR3 | O14843 | 82 | 81 | 9 | 0.85 | 27 | 1.00 | 4 | EC50 81, IC50 1 |
| 212 | VIPR2 | P41587 | 80 | 78 | 9 | 0.75 | 16 | 0.60 | 5 | EC50 48, IC50 32 |
| 213 | RXFP4 | Q8TDU9 | 80 | 53 | 11 | 0.72 | 25 | 0.67 | 6 | EC50 46, Ki 27, IC50 7 |
| 214 | NPSR1 | Q6W5P4 | 79 | 78 | 9 | 0.69 | 36 | not scored | IC50 77, EC50 1, Ki 1 | |
| 215 | GPR39 | O43194 | 77 | 77 | 8 | 0.79 | 28 | not scored | EC50 77 | |
| 216 | GPR132 | Q9UNW8 | 76 | 76 | 8 | 0.56 | 16 | not scored | IC50 42, EC50 34 | |
| 217 | TSHR | P16473 | 75 | 75 | 8 | 0.33 | 6 | 1.00 | 4 | IC50 52, EC50 23 |
| 218 | CCR7 | P32248 | 75 | 71 | 9 | 0.88 | 8 | 1.00 | 4 | IC50 60, Ki 13, EC50 1, Kd 1 |
| 219 | OXER1 | Q8TDS5 | 70 | 69 | 8 | 0.79 | 28 | not scored | IC50 63, EC50 7 | |
| 220 | LHCGR | P22888 | 68 | 66 | 7 | 0.91 | 11 | 1.00 | 1 | EC50 35, IC50 32, Ki 1 |
| 221 | GPR4 | P46093 | 67 | 67 | 8 | 0.89 | 28 | not scored | IC50 67 | |
| 222 | P2RY10 | O00398 | 57 | 57 | 6 | 0.80 | 15 | 0.88 | 8 | EC50 57 |
| 223 | GPR27 | Q9NS67 | 55 | 55 | 6 | 0.60 | 15 | not scored | EC50 55 | |
| 224 | P2RY11 | Q96G91 | 49 | 47 | 5 | 0.67 | 3 | 0.67 | 3 | EC50 28, Ki 15, IC50 6 |
| 225 | GPR12 | P47775 | 47 | 47 | 5 | 0.70 | 10 | 1.00 | 10 | IC50 47 |
| 226 | CCR10 | P46092 | 46 | 46 | 5 | 0.50 | 10 | 1.00 | 7 | IC50 46 |
| 227 | VIPR1 | P32241 | 44 | 41 | 5 | 0.50 | 4 | 0.63 | 40 | EC50 33, IC50 10, Ki 1 |
| 228 | ADGRD1 | Q6QNK2 | 38 | 38 | 4 | 0.33 | 6 | not scored | EC50 38 | |
| 229 | FZD7 | O75084 | 36 | 32 | 5 | 0.83 | 6 | 1.00 | 1 | Kd 32, IC50 4 |
| 230 | MC2R | Q01718 | 35 | 28 | 3 | 1.00 | 1 | not scored | Ki 21, Kb 13, IC50 1 | |
| 231 | MRGPRD | Q8TDS7 | 34 | 34 | 4 | not scored | not scored | IC50 34 | ||
| 232 | TRHR | P34981 | 32 | 16 | 4 | 1.00 | 2 | not scored | Ki 16, EC50 16 | |
| 233 | ADGRF1 | Q5T601 | 24 | 23 | 2 | not scored | 0.71 | 21 | IC50 17, EC50 7 | |
| 234 | OR51E2 | Q9H255 | 22 | 22 | 2 | 0.00 | 1 | not scored | EC50 21, IC50 1 | |
| 235 | LPAR4 | Q99677 | 20 | 20 | 2 | 1.00 | 1 | 0.50 | 6 | EC50 14, IC50 4, Ki 2 |
| 236 | C5AR2 | Q9P296 | 15 | 14 | 3 | not scored | 0.00 | 1 | IC50 10, EC50 2, Kd 2, Ki 1 | |
| 237 | TAS2R46 | P59540 | 14 | 13 | 2 | 1.00 | 1 | 1.00 | 1 | EC50 8, IC50 6 |
| 238 | nan | P31645 | 14 | 14 | 2 | not scored | not scored | Ki 14 | ||
| 239 | TAS2R31 | P59538 | 13 | 13 | 1 | not scored | not scored | EC50 7, IC50 6 | ||
| 240 | P2RY13 | Q9BPV8 | 13 | 13 | 2 | 1.00 | 1 | not scored | EC50 7, IC50 6 | |
| 241 | SCTR | P47872 | 12 | 11 | 1 | not scored | not scored | EC50 11, Ki 1 | ||
| 242 | LPAR6 | P43657 | 11 | 11 | 1 | not scored | 0.80 | 5 | EC50 11 | |
| 243 | TAS2R38 | P59533 | 11 | 11 | 1 | not scored | not scored | EC50 11 | ||
| 244 | GPR68 | Q15743 | 11 | 11 | 1 | not scored | not scored | EC50 9, IC50 2 | ||
| 245 | nan | Q5BJF2 | 11 | 11 | 1 | not scored | not scored | Ki 11 | ||
| 246 | TAS2R16 | Q9NYV7 | 10 | 9 | 1 | not scored | not scored | EC50 9, IC50 1 | ||
| 247 | CMKLR2 | P46091 | 8 | 7 | 1 | not scored | not scored | EC50 6, Ki 2 | ||
| 248 | PROKR2 | Q8NFJ6 | 7 | 7 | 1 | not scored | not scored | Ki 7 | ||
| 249 | OXGR1 | Q96P68 | 7 | 7 | 1 | not scored | 1.00 | 1 | IC50 7 | |
| 250 | GABBR1 | Q9UBS5 | 7 | 6 | 1 | not scored | not scored | EC50 5, Ki 1, IC50 1 | ||
| 251 | ACKR2 | O00590 | 6 | 5 | 1 | not scored | 1.00 | 1 | EC50 5, IC50 1 | |
| 252 | TAS2R10 | Q9NYW0 | 5 | 5 | 1 | not scored | 1.00 | 1 | EC50 5 | |
| 253 | FZD1 | Q9UP38 | 4 | 4 | 1 | not scored | 1.00 | 1 | Kd 2, IC50 1, EC50 1 | |
| 254 | nan | Q12809 | 4 | 4 | 0 | not scored | not scored | IC50 4 | ||
| 255 | TAS2R60 | P59551 | 3 | 3 | 0 | not scored | not scored | EC50 3 | ||
| 256 | TAS2R9 | Q9NYW1 | 3 | 3 | 0 | not scored | not scored | EC50 3 | ||
| 257 | TAS2R4 | Q9NYW5 | 3 | 3 | 0 | not scored | not scored | EC50 3 | ||
| 258 | TAS2R1 | Q9NYW7 | 3 | 3 | 0 | not scored | not scored | EC50 3 | ||
| 259 | MAS1 | P04201 | 2 | 2 | 0 | not scored | not scored | IC50 2 | ||
| 260 | TAS2R41 | P59536 | 2 | 2 | 0 | not scored | not scored | EC50 2 | ||
| 261 | TAS2R43 | P59537 | 2 | 2 | 0 | not scored | not scored | EC50 2 | ||
| 262 | FZD2 | Q14332 | 2 | 2 | 0 | not scored | not scored | IC50 1, EC50 1 | ||
| 263 | TAS2R13 | Q9NYV9 | 2 | 2 | 0 | not scored | not scored | EC50 2 | ||
| 264 | TAAR5 | O14804 | 1 | 1 | 0 | not scored | not scored | EC50 1 | ||
| 265 | GPR37L1 | O60883 | 1 | 1 | 0 | not scored | not scored | IC50 1 | ||
| 266 | ADGRE5 | P48960 | 1 | 1 | 0 | not scored | not scored | Kd 1 | ||
| 267 | GPR15 | P49685 | 1 | 1 | 0 | not scored | not scored | EC50 1 | ||
| 268 | TAS2R39 | P59534 | 1 | 1 | 0 | not scored | not scored | EC50 1 | ||
| 269 | TAS2R40 | P59535 | 1 | 1 | 0 | not scored | not scored | EC50 1 | ||
| 270 | TAS2R45 | P59539 | 1 | 1 | 0 | not scored | not scored | EC50 1 | ||
| 271 | TAS2R30 | P59541 | 1 | 1 | 0 | not scored | not scored | EC50 1 | ||
| 272 | TAS2R19 | P59542 | 1 | 1 | 0 | not scored | not scored | EC50 1 | ||
| 273 | TAS2R20 | P59543 | 1 | 1 | 0 | not scored | not scored | EC50 1 | ||
| 274 | TAS2R50 | P59544 | 1 | 1 | 0 | not scored | not scored | EC50 1 | ||
| 275 | GHRHR | Q02643 | 1 | 1 | 0 | not scored | not scored | IC50 1 | ||
| 276 | OR10J3 | Q5JRS4 | 1 | 1 | 0 | not scored | not scored | Kd 1 | ||
| 277 | TAS2R42 | Q7RTR8 | 1 | 1 | 0 | not scored | not scored | EC50 1 | ||
| 278 | GPR135 | Q8IZ08 | 1 | 1 | 0 | not scored | not scored | EC50 1 | ||
| 279 | LGR4 | Q9BXB1 | 1 | 1 | 0 | not scored | not scored | EC50 1 | ||
| 280 | TAS2R7 | Q9NYW3 | 1 | 1 | 0 | not scored | not scored | EC50 1 | ||
| 281 | TAS2R5 | Q9NYW4 | 1 | 1 | 0 | not scored | not scored | EC50 1 | ||
| 282 | TAS2R3 | Q9NYW6 | 1 | 1 | 0 | not scored | not scored | EC50 1 | ||
| 283 | GPR143 | P51810 | 0 | 0 | 1 | not scored | not scored | |||
| 284 | MRGPRX3 | Q96LB0 | 0 | 0 | 1 | not scored | not scored |