GPCR Foundation Model

Targets in the training set

284 targets, 350,097 fitting measurements and 38,916 held-out measurements. Generated from the measurement files the models were built from.

Gene symbols link to GeneCards and accessions to UniProt. The two accuracy columns are that target's own held-out accuracy, with the number of comparisons it rests on beside it. A target with few comparisons can read 0.00 or 1.00 and neither means much. Targets the model was not scored on say so.

Accuracy depends on the cutoff you are willing to act at. The figures below default to answering every comparison, which is a strength cutoff of 0.50. Raise the cutoff and accuracy rises while the number of comparisons that clear it falls, at very different rates from one target to the next.

Every column heading sorts, except endpoints. Click once for descending, again for ascending. The default is fitting measurements, largest first.

0.50
answer everything
0.600.700.80 0.90
strictest

#▾ Gene▾ Accession▾ Fit measurements▾ Fit ligands▾ Held-out▾ Potency accuracy▾ Potency n▾ Selectivity accuracy▾ Selectivity n▾ Endpoints
1DRD2P1441610,9819,9821,2060.7413,1620.812,454Ki 8836, IC50 1100, EC50 802, Kb 152, Kd 91
2CNR2P3497210,3218,9861,1610.7613,6320.90772Ki 4578, EC50 4103, IC50 1616, Kb 12, Kd 12
3OPRM1P3537210,0958,5931,1260.7713,3200.811,561Ki 5841, EC50 2405, IC50 1773, Kb 43, Kd 33
4CNR1P215549,4098,2841,0450.7912,8220.90785Ki 3703, EC50 3522, IC50 1942, Kd 168, Kb 74
5HCRTR2O436148,1737,8619150.7713,8220.90755IC50 5028, Ki 2169, EC50 800, Kd 129, Kb 47
6ADORA2AP292747,9797,5598880.769,7460.831,162Ki 5962, IC50 1614, EC50 308, Kd 77, Kb 18
7OPRK1P411457,6996,5498720.7614,4380.821,272Ki 4124, IC50 1849, EC50 1656, Kb 51, Kd 19
8HCRTR1O436137,3076,9898190.7910,2710.89757IC50 4800, Ki 2078, EC50 262, Kd 134, Kb 33
9HTR2AP282237,2156,4648070.7314,2870.792,017Ki 5000, IC50 1232, EC50 940, Kb 39, Kd 4
10OPRD1P411436,9825,8197670.7813,5650.881,167Ki 4148, EC50 1439, IC50 1316, Kd 41, Kb 38
11DRD3P354626,6426,0747550.757,7950.781,896Ki 5700, EC50 493, IC50 396, Kb 30, Kd 23
12HTR1AP089086,4885,8687150.7310,7160.761,670Ki 4894, EC50 836, IC50 650, Kd 60, Kb 48
13ADORA1P305426,0825,6996810.738,5000.831,052Ki 4733, IC50 757, EC50 434, Kd 150, Kb 8
14ADORA3P0DMS85,9715,4806700.768,3780.821,069Ki 4714, IC50 907, EC50 250, Kd 68, Kb 32
15PTGDR2Q9Y5Y45,9515,6296520.739,5040.9565IC50 3661, Ki 1725, EC50 554, Kb 6, Kd 5
16HTR6P504065,1334,3435670.769,3950.741,001Ki 3769, IC50 887, Kb 272, EC50 135, Kd 70
17HRH3Q9Y5N15,0534,3005470.748,0360.84279Ki 3664, IC50 727, EC50 339, Kd 251, Kb 72
18HTR2CP283354,7884,2765380.7213,7740.801,522Ki 2712, EC50 1061, IC50 1005, Kb 8, Kd 2
19ADORA2BP292754,7454,5325190.809,5180.91719Ki 2536, IC50 1744, EC50 385, Kb 43, Kd 37
20LPAR1Q926334,5224,3965070.715,5460.8336IC50 3903, EC50 449, Ki 125, Kb 39, Kd 6
21MC4RP322454,3713,3934740.7914,3620.80446Ki 1852, EC50 1454, IC50 1025, Kd 27, Kb 13
22CRHR1P349984,0653,8264520.785,0530.8211IC50 2487, Ki 1465, EC50 93, Kd 20
23S1PR1P214533,9123,5564410.779,3560.94384EC50 2502, IC50 1271, Ki 129, Kd 9, Kb 1
24MCHR1Q997053,9103,6674380.739,8050.8257IC50 2306, Ki 1483, EC50 61, Kb 57, Kd 3
25GRM5P415943,6283,1864100.7510,9510.8488IC50 1894, EC50 1198, Ki 525, Kb 9, Kd 2
26DRD4P219173,4963,0593850.726,4860.801,080Ki 2758, IC50 369, EC50 354, Kd 12, Kb 3
27CHRM1P112293,4643,2493920.7413,8840.75903Ki 1501, EC50 886, IC50 860, Kb 148, Kd 69
28APLNRP354143,3583,1963710.735,2530.6644EC50 2984, Ki 240, IC50 133, Kd 1
29HTR7P349693,3453,1653670.736,2940.761,025Ki 2631, IC50 416, EC50 231, Kb 58, Kd 9
30GLP1RP432203,0992,9243450.814,9170.7876EC50 2813, IC50 231, Ki 45, Kd 10
31OPRL1P411463,0842,6843420.767,8320.90370Ki 2003, IC50 647, EC50 372, Kb 51, Kd 11
32CHRM3P203093,0832,8973480.829,1970.76859Ki 1887, IC50 942, EC50 167, Kd 87
33HRH4Q9H3N83,0622,6973310.755,4270.85215Ki 1673, EC50 1014, IC50 188, Kd 131, Kb 56
34MRGPRX2Q96LB12,8112,7853130.832,7271.004IC50 2496, EC50 289, Kd 26
35CHRM2P081722,7872,5323170.808,1800.78853Ki 1598, IC50 601, EC50 272, Kb 178, Kd 138
36HRH1P353672,7842,6153130.775,6760.76769Ki 1506, EC50 664, IC50 391, Kd 164, Kb 59
37ADRB2P075502,7282,3583000.8110,0650.77476EC50 1217, IC50 675, Ki 665, Kd 169, Kb 2
38TACR1P251032,6162,4952930.809,3390.78162IC50 1643, Ki 860, Kd 96, EC50 15, Kb 2
39HTR2BP415952,5652,1692880.747,2080.741,146Ki 1669, EC50 526, IC50 345, Kb 24, Kd 1
40FFAR1O148422,5502,3992840.724,8320.9432EC50 2320, Ki 126, IC50 94, Kd 10
41S1PR3Q995002,4502,4112720.835,9460.94359EC50 1617, IC50 820, Kd 8, Ki 5
42GHSRQ928472,3461,9252610.7210,4620.867IC50 879, EC50 792, Ki 603, Kb 69, Kd 3
43CHRM4P081732,3022,1592590.777,9450.78691Ki 1312, EC50 656, IC50 300, Kb 27, Kd 7
44CCR5P516812,2612,2302570.775,0730.7356IC50 2050, Ki 142, EC50 55, Kd 14
45FPR2P250902,1542,0972370.786,9690.8686EC50 1326, IC50 462, Kd 339, Ki 27
46GRM2Q144162,1221,8952280.769,8840.6972EC50 939, IC50 921, Ki 205, Kd 44, Kb 13
47CCR2P415972,0701,9852270.735,1350.9521IC50 1754, Ki 290, Kd 17, EC50 9
48ADRA1AP353482,0441,9312240.805,7570.83774Ki 1414, IC50 309, EC50 290, Kd 18, Kb 13
49CHRM5P089122,0231,9352250.758,3140.75621IC50 911, Ki 896, EC50 213, Kd 3
50AVPR1AP372881,9781,6912200.787,2010.83224Ki 1049, IC50 690, EC50 214, Kb 17, Kd 8
51DRD1P217281,9471,7502140.765,3460.75782Ki 1423, EC50 265, IC50 218, Kd 30, Kb 11
52ADRB1P085881,8491,7092040.786,2500.81527EC50 760, IC50 588, Ki 403, Kd 97, Kb 1
53GPR17Q133041,8261,8132070.793,0930.6916IC50 1532, Kb 212, EC50 67, Ki 14, Kd 1
54GPR119Q8TDV51,7371,6781900.744,6610.5024EC50 1656, Ki 47, IC50 34
55CXCR3P496821,7091,6791890.765,2460.4719IC50 1405, Ki 266, EC50 34, Kd 4
56CCKBRP322391,6961,5531790.826,2620.8547IC50 1131, Ki 452, EC50 106, Kd 7
57ADRA1BP353681,6881,6161840.764,8120.78613Ki 1310, EC50 213, IC50 150, Kd 10, Kb 5
58GRM4Q148331,6551,6001900.774,9720.7879EC50 1487, IC50 85, Ki 70, Kb 13
59ADRB3P139451,6531,5391880.745,6310.79392EC50 1174, Ki 340, IC50 82, Kd 57
60P2RY1P479001,6171,1421810.704,3600.7114Ki 961, IC50 587, EC50 62, Kd 6, Kb 1
61GNRHRP309681,6141,5151790.787,0021.002IC50 912, Ki 664, Kd 35, EC50 2, Kb 1
62EDNRAP251011,5851,5161730.805,0790.70178IC50 1278, Ki 227, Kb 65, EC50 11, Kd 4
63SSTR4P313911,5841,3361800.765,3080.82253EC50 604, IC50 532, Ki 418, Kd 30
64HTR1DP282211,5691,3831710.805,6740.77597Ki 1081, IC50 310, EC50 166, Kb 9, Kd 3
65ADRA1DP251001,5671,4331700.754,8880.80605Ki 1139, IC50 219, EC50 204, Kb 5
66MC1RQ017261,5491,0951660.814,9220.83249EC50 737, Ki 482, IC50 326, Kd 4
67MC5RP330321,5161,2691670.832,7060.76257IC50 771, Ki 421, EC50 320, Kd 4
68PTGER4P354081,4981,2651660.794,6430.93187IC50 661, Ki 534, EC50 252, Kb 44, Kd 7
69MC3RP419681,4971,0751600.814,1760.83355Ki 607, EC50 502, IC50 368, Kd 20
70GCGRP478711,4761,4201660.804,7250.8848IC50 782, EC50 372, Ki 273, Kb 49
71SSTR2P308741,4611,4271630.853,1330.82240Ki 526, IC50 457, EC50 443, Kd 35
72AGTR1P305561,4581,4071640.864,9840.67121IC50 1062, Ki 200, EC50 164, Kd 24, Kb 8
73ADRA2AP089131,4421,1781620.785,3870.74811Ki 910, IC50 273, EC50 186, Kb 67, Kd 6
74ACKR3P251061,4331,4171620.755,0681.0012IC50 722, EC50 625, Ki 83, Kd 3
75HTR1BP282221,4171,3191560.805,1740.79551Ki 1013, IC50 280, EC50 111, Kd 7, Kb 6
76FFAR4Q5NUL31,4121,4101570.784,1650.8843EC50 1400, IC50 12
77TACR3P293711,4031,1591560.794,5020.7898Ki 806, IC50 463, EC50 114, Kb 10, Kd 10
78P2RY12Q9H2441,3831,2081590.774,9770.805IC50 701, Ki 607, EC50 68, Kb 4, Kd 3
79CXCR2P250251,3291,2911540.774,4780.8491IC50 1094, Ki 215, Kd 18, EC50 2
80CXCR4P610731,3191,2001490.714,7930.8527IC50 1094, EC50 204, Ki 13, Kb 4, Kd 4
81NPY5RQ157611,3131,2461430.754,6500.9355IC50 714, Ki 563, EC50 32, Kb 4
82NPY1RP259291,3031,1781410.813,3770.70124Ki 602, IC50 481, EC50 142, Kb 58, Kd 20
83MTNR1AP480391,2881,0971450.794,7280.74157Ki 891, IC50 204, EC50 168, Kb 23, Kd 2
84OXTRP305591,2421,1241320.803,2080.87138Ki 635, EC50 360, IC50 214, Kd 33
85CRHR2Q133241,2331,2281371.002800.888IC50 1219, Ki 9, EC50 5
86TBXA2RP217311,2191,1781380.832,9890.8896IC50 560, Ki 412, Kd 204, EC50 41, Kb 2
87F2RL3Q96RI01,2181,1321330.794,4921.007IC50 793, EC50 422, Kd 3
88GPBAR1Q8TDU61,1981,1941330.724,8330.001EC50 1166, IC50 32
89EDNRBP245301,1691,1401270.824,8320.86118IC50 981, Ki 177, Kd 5, Kb 4, EC50 2
90CALCRLQ166021,1528201330.854,158not scoredKi 580, IC50 547, EC50 12, Kd 7, Kb 6
91MTNR1BP492861,1459601370.774,6200.84121Ki 858, EC50 165, IC50 86, Kb 33, Kd 3
92SSTR3P327451,1389781280.842,3100.80228IC50 531, Ki 361, EC50 176, Kd 70
93GRM1Q132551,1381,0401290.843,8040.82102IC50 781, EC50 255, Ki 88, Kb 14
94SSTR5P353461,1291,0861260.853,3100.85239IC50 668, Ki 360, EC50 68, Kd 33
95C5AR1P217301,1251,1021290.824,4910.605IC50 1022, EC50 49, Ki 41, Kb 10, Kd 3
96PTGER3P431151,1189671190.832,5010.87121IC50 501, Ki 485, EC50 121, Kb 11
97TAAR1Q96RJ01,1136991270.623,8451.001EC50 659, IC50 408, Ki 46
98AVPR2P305181,1071,0381230.822,5340.84167Ki 470, IC50 367, EC50 261, Kd 9
99TACR2P214521,1051,0431240.873,9370.65267Ki 805, IC50 285, Kd 9, EC50 5, Kb 1
100NPY2RP491461,0989791210.902,5200.71111IC50 532, Ki 279, EC50 271, Kd 15, Kb 1
101PTGER2P431161,0819681170.811,6820.90157Ki 380, EC50 323, IC50 196, Kb 175, Kd 7
102CCR3P516771,0691,0591180.823,9360.9122IC50 686, Ki 373, EC50 5, Kb 3, Kd 2
103ADRA2CP188251,0648211210.713,3490.73727Ki 705, EC50 148, IC50 140, Kb 70, Kd 1
104PTGER1P349951,0449231210.792,9930.85101IC50 607, Ki 371, EC50 42, Kd 14, Kb 10
105BDKRB1P466631,0418051140.743,0730.789Ki 637, IC50 398, Kd 2, Kb 2, EC50 2
106GPR6P460951,0401,0351170.813,5451.0010IC50 675, EC50 360, Ki 4, Kd 1
107FPR1P214621,0069751100.711,9440.8463EC50 503, Ki 255, IC50 206, Kd 42
108F2RP251169629101100.823,7761.006IC50 780, EC50 95, Ki 73, Kd 14
109HTR4Q136399477581000.782,2010.86101Ki 459, EC50 386, IC50 87, Kb 12, Kd 3
110GPR55Q9Y2T69388791080.792,5670.7672IC50 557, EC50 374, Kb 4, Kd 3
111GPR84Q9NQS59078431020.792,339not scoredIC50 564, EC50 267, Ki 70, Kd 4, Kb 2
112HRH2P25021905744990.821,5510.74449Ki 574, EC50 136, IC50 118, Kd 60, Kb 17
113S1PR2O951369048881020.901,4770.88142IC50 611, EC50 226, Kd 66, Ki 1
114CCR4P51679891821960.832,4790.7512IC50 751, Ki 90, Kd 41, EC50 9
115CCR1P32246889842960.783,0940.8055IC50 722, Ki 148, EC50 18, Kd 1
116ADRA2BP180898846881010.682,2170.71673Ki 603, IC50 160, EC50 84, Kb 36, Kd 1
117GPR35Q9HC97882570990.851,6210.8366EC50 422, IC50 400, Ki 56, Kd 4
118PTGDRQ13258881796910.881,2450.92128IC50 440, Ki 325, Kb 58, EC50 57, Kd 1
119CCR6P51684863859980.884,0180.7621IC50 858, Ki 4, EC50 1
120HCAR2Q8TDS4855663980.822,4620.8312EC50 562, IC50 261, Ki 32
121AVPR1BP47901815805920.861,4610.95116IC50 395, Ki 223, EC50 192, Kd 5
122SSTR1P30872807797900.861,3250.88232IC50 504, Ki 238, Kd 50, EC50 15
123NTSR1P30989791699800.761,2810.6659EC50 511, Ki 152, IC50 115, Kd 13
124FFAR2O15552790768870.741,6571.004EC50 588, IC50 178, Ki 24
125S1PR4O95977789778880.811,6610.87161IC50 439, EC50 339, Kd 8, Ki 2, Kb 1
126SMOQ99835775752880.793,129not scoredIC50 729, EC50 21, Ki 20, Kd 5
127AGTR2P50052761752850.802,2160.9841IC50 544, Ki 217
128HTR5AP47898741707810.841,3410.78403Ki 451, EC50 242, IC50 46, Kd 2
129UTS2RQ9UKP6694618740.80826not scoredKi 292, EC50 218, IC50 179, Kd 5
130CCKARP32238686470690.877240.7980IC50 318, EC50 191, Ki 176, Kd 1
131PTGIRP43119628583700.795070.8770Ki 256, IC50 166, EC50 162, Kb 44
132PTAFRP25105625616680.802,0181.001IC50 602, Ki 22, Kd 1
133BDKRB2P30411625537690.848580.7345Ki 303, IC50 225, Kd 95, EC50 2
134S1PR5Q9H228619605680.781,1290.82151EC50 354, IC50 252, Kd 8, Ki 5
135DRD5P21918594581660.811,4520.80379Ki 533, EC50 40, IC50 18, Kd 3
136CX3CR1P49238594589650.801,1520.7438IC50 469, EC50 70, Ki 55
137CASRP41180592591660.801,0671.001IC50 360, EC50 232
138PTGFRP43088567555630.831,1290.9158IC50 418, Ki 86, EC50 61, Kb 2
139MLNRO43193548484640.706081.003EC50 290, Ki 160, IC50 98
140LTB4RQ15722530491590.77542not scoredIC50 249, EC50 152, Ki 123, Kb 5, Kd 1
141BRS3P32247527363530.797040.717EC50 328, IC50 178, Ki 21
142NPBWR1P48145506499560.831,2750.6724IC50 460, EC50 46
143CALCRP30988480355480.86703not scoredEC50 342, IC50 125, Ki 13
144GPR183P32249464463520.821,0890.6330IC50 455, EC50 8, Kd 1
145FPR3P25089456456510.871,0170.8066EC50 419, IC50 37
146GPR88Q9GZN0449444490.801,162not scoredEC50 443, Ki 5, Kd 1
147P2RY2P41231442434500.764240.7340EC50 248, IC50 132, Kd 40, Ki 22
148NPY4RP50391431275520.844250.9155Ki 215, EC50 135, IC50 44, Kb 32, Kd 5
149GPR139Q6DWJ6420336440.79592not scoredEC50 334, Ki 86
150CMKLR1Q99788415385460.912571.003IC50 332, EC50 82, Ki 1
151GIPRP48546406405450.842370.8730EC50 263, IC50 140, Ki 3
152P2RY14Q15391404377460.784880.8817IC50 321, EC50 47, Ki 31, Kd 4, Kb 1
153CXCR1P25024386377420.833591.0037IC50 290, Ki 91, Kd 4, EC50 1
154P2RY6Q15077375373420.744240.6433EC50 252, IC50 115, Ki 6, Kd 2
155LPAR2Q9HBW0367362410.873720.8432IC50 299, EC50 61, Ki 7
156CCR9P51686359357400.89159not scoredIC50 237, Ki 121, EC50 1
157KISS1RQ969F8357284440.823621.004EC50 186, IC50 94, Ki 77
158GPR52Q9Y2T5332332370.86486not scoredEC50 308, IC50 24
159GRM3Q14832329242390.792230.7158IC50 144, EC50 109, Ki 76
160PRLHRP49683314231350.80204not scoredKi 144, IC50 86, EC50 84
161HTR1EP28566309287350.861760.84282Ki 237, IC50 40, EC50 32
162GRM7Q14831302288330.791230.9735IC50 163, EC50 122, Ki 17
163PTH1RQ03431298282320.88199not scoredEC50 213, IC50 55, Ki 24, Kd 6
164TAS2R8Q9NYW2290290320.82491not scoredIC50 289, EC50 1
165PROKR1Q8TCW9282282310.69463not scoredIC50 279, Ki 3
166CXCR6O00574280278310.94212not scoredIC50 278, EC50 1, Kd 1
167MRGPRX4Q96LA9278278310.79248not scoredIC50 278
168LPAR3Q9UBY5271232280.811400.7520IC50 147, EC50 65, Ki 59
169C3AR1Q16581261207290.632050.754IC50 162, EC50 98, Kd 1
170CYSLTR1Q9Y271250241300.842780.4238IC50 217, Ki 12, EC50 12, Kd 9
171CCR8P51685246236270.761720.254IC50 162, Ki 68, EC50 16
172GRPRP30550240232260.832480.717IC50 184, Ki 47, EC50 8, Kb 1
173GALR3O60755239239260.64220not scoredIC50 211, Ki 24, Kd 4
174GPR18Q14330238190290.901340.8918IC50 128, EC50 108, Kd 1, Kb 1
175P2RY4P51582229228250.831390.7431EC50 148, IC50 80, Kb 1
176RXFP1Q9HBX9229226250.822971.002EC50 218, IC50 6, Ki 5
177F2RL1P55085218216250.601241.001EC50 113, IC50 103, Ki 2
178NPFFR2Q9Y5X5201175200.821260.8432Ki 120, EC50 66, IC50 8, Kd 7
179GPR142Q7Z601199199220.77149not scoredEC50 156, IC50 43
180HTR1FP30939198172190.62580.76109Ki 125, EC50 59, IC50 14
181GRM8O00222196186230.73910.8753EC50 134, IC50 42, Ki 19, Kd 1
182NTSR2O95665194184200.64720.8816Ki 116, EC50 49, IC50 26, Kd 3
183GPR3P46089187184200.79781.0010IC50 142, EC50 43, Kd 1, Ki 1
184NPFFR1Q9GZQ6184160210.741080.8825Ki 116, EC50 50, Kd 9, IC50 8, Kb 1
185HCAR1Q9BXC0180180200.771111.002EC50 180
186NMBRP28336174167190.81590.676Ki 100, IC50 64, EC50 8, Kb 2
187NMUR2Q9GZQ4163119170.79720.6913EC50 113, IC50 43, Ki 3, Kd 2, Kb 2
188ADCYAP1R1P4158616295180.83600.002IC50 79, EC50 65, Ki 15, Kd 3
189QRFPRQ96P65161128160.86491.002EC50 85, IC50 71, Ki 5
190GRM6O15303157148180.76710.8642EC50 98, IC50 36, Ki 23
191LPAR5Q9H1C0157156170.851300.7311IC50 142, EC50 14, Ki 1
192MRGPRX1Q96LB2144144160.81631.002EC50 117, IC50 27
193MCHR2Q969V1142141160.85340.899Ki 86, IC50 56
194RXFP3Q9NSD7142118160.86360.676EC50 66, IC50 41, Ki 35
195CCRL2O00421140140160.761191.001IC50 140
196TAS2R14Q9NYV8139138150.7769not scoredIC50 105, EC50 34
197GPR34Q9UPC5133133151.00131.003IC50 93, EC50 40
198NMUR1Q9HB8913190140.81420.6913EC50 81, IC50 43, Ki 3, Kd 2, Kb 2
199GALR2O43603128125140.58430.6444IC50 78, Ki 32, EC50 11, Kd 7
200HCAR3P49019114113130.85750.758EC50 110, IC50 4
201FSHRP23945111111120.69321.003EC50 56, IC50 55
202GPER1Q99527109105130.29280.001IC50 100, EC50 5, Ki 3, Kd 1
203GLP2RO95838108108120.80550.9212EC50 100, IC50 8
204LTB4R2Q9NPC110899110.8445not scoredEC50 67, IC50 37, Kd 3, Ki 1
205CYSLTR2Q9NS75108105120.88520.8324IC50 97, EC50 10, Ki 1
206GPR65Q8IYL9106106120.89450.7423IC50 103, EC50 3
207SUCNR1Q9BXA510191110.71241.001IC50 70, EC50 19, Ki 9, Kd 3
208GALR1P472119995110.72250.758IC50 58, Ki 34, Kd 7
209GPR174Q9BXC19388110.69320.805EC50 88, IC50 5
210CXCR5P323028988100.78450.388IC50 87, EC50 2
211FFAR3O14843828190.85271.004EC50 81, IC50 1
212VIPR2P41587807890.75160.605EC50 48, IC50 32
213RXFP4Q8TDU98053110.72250.676EC50 46, Ki 27, IC50 7
214NPSR1Q6W5P4797890.6936not scoredIC50 77, EC50 1, Ki 1
215GPR39O43194777780.7928not scoredEC50 77
216GPR132Q9UNW8767680.5616not scoredIC50 42, EC50 34
217TSHRP16473757580.3361.004IC50 52, EC50 23
218CCR7P32248757190.8881.004IC50 60, Ki 13, EC50 1, Kd 1
219OXER1Q8TDS5706980.7928not scoredIC50 63, EC50 7
220LHCGRP22888686670.91111.001EC50 35, IC50 32, Ki 1
221GPR4P46093676780.8928not scoredIC50 67
222P2RY10O00398575760.80150.888EC50 57
223GPR27Q9NS67555560.6015not scoredEC50 55
224P2RY11Q96G91494750.6730.673EC50 28, Ki 15, IC50 6
225GPR12P47775474750.70101.0010IC50 47
226CCR10P46092464650.50101.007IC50 46
227VIPR1P32241444150.5040.6340EC50 33, IC50 10, Ki 1
228ADGRD1Q6QNK2383840.336not scoredEC50 38
229FZD7O75084363250.8361.001Kd 32, IC50 4
230MC2RQ01718352831.001not scoredKi 21, Kb 13, IC50 1
231MRGPRDQ8TDS734344not scorednot scoredIC50 34
232TRHRP34981321641.002not scoredKi 16, EC50 16
233ADGRF1Q5T60124232not scored0.7121IC50 17, EC50 7
234OR51E2Q9H255222220.001not scoredEC50 21, IC50 1
235LPAR4Q99677202021.0010.506EC50 14, IC50 4, Ki 2
236C5AR2Q9P29615143not scored0.001IC50 10, EC50 2, Kd 2, Ki 1
237TAS2R46P59540141321.0011.001EC50 8, IC50 6
238nanP3164514142not scorednot scoredKi 14
239TAS2R31P5953813131not scorednot scoredEC50 7, IC50 6
240P2RY13Q9BPV8131321.001not scoredEC50 7, IC50 6
241SCTRP4787212111not scorednot scoredEC50 11, Ki 1
242LPAR6P4365711111not scored0.805EC50 11
243TAS2R38P5953311111not scorednot scoredEC50 11
244GPR68Q1574311111not scorednot scoredEC50 9, IC50 2
245nanQ5BJF211111not scorednot scoredKi 11
246TAS2R16Q9NYV71091not scorednot scoredEC50 9, IC50 1
247CMKLR2P46091871not scorednot scoredEC50 6, Ki 2
248PROKR2Q8NFJ6771not scorednot scoredKi 7
249OXGR1Q96P68771not scored1.001IC50 7
250GABBR1Q9UBS5761not scorednot scoredEC50 5, Ki 1, IC50 1
251ACKR2O00590651not scored1.001EC50 5, IC50 1
252TAS2R10Q9NYW0551not scored1.001EC50 5
253FZD1Q9UP38441not scored1.001Kd 2, IC50 1, EC50 1
254nanQ12809440not scorednot scoredIC50 4
255TAS2R60P59551330not scorednot scoredEC50 3
256TAS2R9Q9NYW1330not scorednot scoredEC50 3
257TAS2R4Q9NYW5330not scorednot scoredEC50 3
258TAS2R1Q9NYW7330not scorednot scoredEC50 3
259MAS1P04201220not scorednot scoredIC50 2
260TAS2R41P59536220not scorednot scoredEC50 2
261TAS2R43P59537220not scorednot scoredEC50 2
262FZD2Q14332220not scorednot scoredIC50 1, EC50 1
263TAS2R13Q9NYV9220not scorednot scoredEC50 2
264TAAR5O14804110not scorednot scoredEC50 1
265GPR37L1O60883110not scorednot scoredIC50 1
266ADGRE5P48960110not scorednot scoredKd 1
267GPR15P49685110not scorednot scoredEC50 1
268TAS2R39P59534110not scorednot scoredEC50 1
269TAS2R40P59535110not scorednot scoredEC50 1
270TAS2R45P59539110not scorednot scoredEC50 1
271TAS2R30P59541110not scorednot scoredEC50 1
272TAS2R19P59542110not scorednot scoredEC50 1
273TAS2R20P59543110not scorednot scoredEC50 1
274TAS2R50P59544110not scorednot scoredEC50 1
275GHRHRQ02643110not scorednot scoredIC50 1
276OR10J3Q5JRS4110not scorednot scoredKd 1
277TAS2R42Q7RTR8110not scorednot scoredEC50 1
278GPR135Q8IZ08110not scorednot scoredEC50 1
279LGR4Q9BXB1110not scorednot scoredEC50 1
280TAS2R7Q9NYW3110not scorednot scoredEC50 1
281TAS2R5Q9NYW4110not scorednot scoredEC50 1
282TAS2R3Q9NYW6110not scorednot scoredEC50 1
283GPR143P51810001not scorednot scored
284MRGPRX3Q96LB0001not scorednot scored